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Viser treff 1-38 av 38

2023
1 Ausbacher, Dominik; Miller, Lindsey A.; Goeres, Darla M.; Stewart, Philip S.; Strøm, Morten Bøhmer; Fallarero, Adyary.
α,α-disubstituted β-amino amides eliminate Staphylococcus aureus biofilms by membrane disruption and biomass removal. Biofilm 2023 ;Volum 6.
UiT Untitled
 
2 von Hofsten, Susannah; Langer, Manuel K; Korelin, Katja; Norvoll Magnussen, Synnøve; Ausbacher, Dominik; Anderssen, Trude; Salo, Tuula; Strøm, Morten B.; Bayer, Annette; Al-Samadi, Ahmed; Berge, Gerd.
Amphipathic barbiturates as marine product mimics with cytolytic and immunogenic effects on head and neck squamous cell carcinoma cell lines. Frontiers in Pharmacology 2023 ;Volum 14.
UiT Untitled
 
2022
3 von Hofsten, Susannah; Paulsen, Marianne Hagensen; Langer, Manuel K; Norvoll Magnussen, Synnøve; Ausbacher, Dominik; Bayer, Annette; Strøm, Morten B.; Berge, Gerd.
A Compound Inspired by Arctic Marine Animals Kills Cancer Cells in vitro and in vivo. IMB Conference 2022; 2022-06-13 - 2022-06-14
UiT Untitled
 
4 von Hofsten, Susannah; Paulsen, Marianne Hagensen; Magnussen, Synnøve; Ausbacher, Dominik; Kranz, Mathias; Bayer, Annette; Strøm, Morten Bøhmer; Berge, Gerd.
The marine natural product mimic MPM-1 is cytolytic and induces DAMP release from human cancer cell lines. Scientific Reports 2022 ;Volum 12.(1)
UiT UNN Untitled
 
2021
5 Paulsen, Marianne Hagensen; Engqvist, Magnus; Ausbacher, Dominik; Anderssen, Trude; Langer, Manuel K-; Haug, Tor; Morello, Glenn Robert; Liikanen, Laura; Blencke, Hans-Matti; Isaksson, Johan; Juskewitz, Eric; Bayer, Annette; Strøm, Morten B..
Amphipathic Barbiturates as Mimics of Antimicrobial Peptides and the Marine Natural Products Eusynstyelamides with Activity against Multi-resistant Clinical Isolates. Journal of Medicinal Chemistry 2021 ;Volum 64.(15) s. 11395-11417
UiT Untitled
 
2020
6 Eksteen, Jacobus Johannes; Ausbacher, Dominik; Vasskog, Terje; Rekdal, Øystein; Svendsen, John Sigurd Mjøen.
Selective intracellular delivery of thiolated cargo to tumor and neovasculature cells using histidine-rich peptides as vectors. ACS Omega 2020 ;Volum 5.(10) s. 4937-4942
UiT NORCE Untitled
 
7 von Hofsten, Susannah; Norvoll Magnussen, Synnøve; Ausbacher, Dominik; Paulsen, Marianne Hagensen; Bayer, Annette; Strøm, Morten B.; Berge, gerd.
The Marine Natural Product Mimic MHP88 Shows Anticancer Activity and has the Potential to Cause Immunogenic Cell Death. EACR-AACR Basic and Translational Research Conference in partnership with ASPIC: Tumor Microenvironment; 2020-03-02 - 2020-03-04
UiT Untitled
 
2019
8 Paulsen, Marianne Hagensen; Ausbacher, Dominik; Bayer, Annette; Engqvist, Magnus; Hansen, Terkel; Haug, Tor; Anderssen, Trude; Andersen, Jeanette hammer; Sollid, Johanna U Ericson; Strøm, Morten B..
Antimicrobial activity of amphipathic α,α-disubstituted β-amino amide derivatives against ESBL–CARBA producing multi-resistant bacteria; effect of halogenation, lipophilicity and cationic character. European Journal of Medicinal Chemistry 2019 ;Volum 183. s. 111671-111682
UiT SNHF Untitled
 
2018
9 Ausbacher, Dominik.
Exploiting innate antimicrobial defenses: Antimicrobial peptides and peptide antibiotics as templates for novel anti-infective therapeutics. Course: Microbial lifestyles and drug discovery of antimicrobials; 2018-04-16 - 2018-05-11
SNHF Untitled
 
10 Paulsen, Marianne Hagensen; Karlsen, Eskil Andre; Ausbacher, Dominik; Anderssen, Trude; Bayer, Annette; Ochtrop, Philipp; Hedberg, Christian; Haug, Tor; Sollid, Johanna U Ericson; Strøm, Morten B..
An amphipathic cyclic tetrapeptide scaffold containing halogenated β2,2-amino acids with activity against multi-resistant bacteria. Journal of Peptide Science 2018 ;Volum 24.(10) s. 1-11
SNHF UiT Untitled
 
2017
11 Ausbacher, Dominik.
Exploiting innate antimicrobial defenses: Antimicrobial peptides and peptide antibiotics as templates for novel anti-infective therapeutics. University of Helsinki - Advanced Course on Microbial Lifestyles and Drug Discovery of Antimicrobials; 2017-05-02 - 2017-05-19
SNHF Untitled
 
12 Ausbacher, Dominik; Lorenz, Lindsey A.; Pitts, Betsey; Stewart, Philip S.; Goeres, Darla M..
Paired methods to measure biofilm killing and removal: a case study with Penicillin G treatment of Staphylococcus aureus biofilm. Letters in Applied Microbiology 2017 ;Volum 66.(3) s. 231-237
UiT Untitled
 
2016
13 Ausbacher, Dominik.
Exploiting innate antimicrobial defenses: Antimicrobial peptides and peptide antibiotics as templates for novel anti-infective therapeutics. University of Helsinki - Advanced Course on Microbial Lifestyles and Drug Discovery of Antimicrobials; 2016-04-26 - 2016-05-27
UiT Untitled
 
14 Ausbacher, Dominik; Lorenz, Lindsey A.; Goeres, Darla M.; Stewart, Philip S.; Strøm, Morten B.; Vuorela, Pia M.; Fallarero, Adyary.
Antimicrobial β2,2-amino acid derivatives eliminate Staphylococcus aureus biofilms by membrane disruption and biomass removal. Annual DPhG meeting; 2016-10-05 - 2016-10-07
UiT Untitled
 
15 Eksteen, Jacobus Johannes; Ausbacher, Dominik; Simon-Santamaria, Jaione; Stiberg, Trine; Cavalcanti Jacobsen, Cristiane de Albuquerque; Wushur, Imin; Svendsen, John Sigurd Mjøen; Rekdal, Øystein.
Iterative design and in vivo evaluation of an oncolytic antilymphoma peptide. Journal of Medicinal Chemistry 2016 ;Volum 60.(1) s. 146-156
UiT Untitled
 
16 Hanski, Leena; Ausbacher, Dominik; Strøm, Morten B.; Vuorela, Pia M.
Impact of β2,2-amino acid derivatives, a novel class of Chlamydia pneumoniae inhibitors, on bronchial epithelium VEGF production.. Conference on Lung and Respiratory Care; 2016-08-01 - 2016-08-02
UiT Untitled
 
17 Hanski, Leena; Ausbacher, Dominik; Tiirola, Terttu; Strøm, Morten B.; Vuorela, Pia M..
Amphipathic β2,2-Amino Acid Derivatives Suppress Infectivity and Disrupt the Intracellular Replication Cycle of Chlamydia Pneumoniae. PLOS ONE 2016 ;Volum 11.(6)
UiT Untitled
 
18 Paulsen, Marianne H.; Engqvist, Magnus; Ausbacher, Dominik; Strøm, Morten B.; Bayer, Annette.
Efficient and scalable synthesis of α,α-disubstituted β-amino amides. Organic and biomolecular chemistry 2016 ;Volum 14.(31) s. 7570-7578
UiT Untitled
 
2015
19 Ausbacher, Dominik.
Antimicrobial and anticancer β2,2-amino acid derivatives: Peptide mimetics with potential for oral administration. Montana Biofilm Meeting; 2015-07-13 - 2015-07-17
UiT Untitled
 
20 Ausbacher, Dominik.
Exploiting innate antimicrobial defenses: Antimicrobial peptides (AMPs) as templates for novel anti-infective therapeutics. University of Helsinki - Advanced Course on Microbial Lifestyles and Drug Discovery of Antimicrobials; 2015-03-23 - 2015-04-24
UiT Untitled
 
21 Ausbacher, Dominik.
β2,2-amino acid derivatives developed from antimicrobial peptides: Biological activity and mechanism of action studies. Center for Biofilm Engineering - Research Seminar; 2015-04-23 - 2015-04-23
UiT Untitled
 
2014
22 Ausbacher, Dominik; Fallarero, Adyary; Kujala, Janni; Määttänen, Anni; Peltonen, Jouko; Strøm, Morten B.; Vuorela, Pia M..
Staphylococcus aureus biofilm susceptibility to small and potent β2,2-amino acid derivatives. Biofouling (Print) 2014 ;Volum 30.(1) s. 81-93
UiT Untitled
 
23 Ausbacher, Dominik; Hanski, Leena; Tiirola, Terttu; Strøm, Morten B.; Pia, Vuorela.
Anti-Chlamydia pneumoniae activity of β2,2- amino acid derivatives mimicking antimicrobial peptides. Center for Drug Research Seminar; 2014-09-04 - 2014-09-05
UiT Untitled
 
24 Sivertsen, Annfrid; Tørfoss, Veronika; Isaksson, Johan; Ausbacher, Dominik; Anderssen, Trude; Brandsdal, Bjørn Olav; Havelkova, Martina; Skjørholm, Anne Elisabeth; Strøm, Morten B..
Anticancer potency of small linear and cyclic tetrapeptides and pharmacokinetic investigations of peptide binding to human serum albumin. Journal of Peptide Science 2014 ;Volum 20.(4) s. 279-291
UiT Untitled
 
2013
25 Fallarero, Adyary; Skogman, Malena; Moreira, Vânia; Manner, Suvi; Ausbacher, Dominik; Leino, Reko; Strøm, Morten B.; Yli-Kauhaluoma, Jari; Vuorela, Pia.
The challenges of discovering new anti-biofilm probes from a high-throughput screening (HTS) perspective. 3rd European Congress on Microbial Biofilms - Basic and Clinical Aspects; 2013-09-09 - 2013-09-12
UiT Untitled
 
2012
26 Ausbacher, Dominik; Kujala, Janni; Vuorela, Pia M.; Strøm, Morten B.; Fallarero, Adyary.
Control of Staphylococcus aureus biofilm with highly active β2,2-amino acid derivatives. 3rd International Symposium on Antimicrobial Peptides; 2012-06-13 - 2012-06-15
UiT Untitled
 
27 Ausbacher, Dominik; Svineng, Gunbjørg; Hansen, Terkel; Strøm, Morten B..
Anticancer mechanisms of action of two small amphipathic beta(2,2)-amino acid derivatives derived from antimicrobial peptides. Biochimica et Biophysica Acta - Biomembranes 2012 ;Volum 1818.(11) s. 2917-2925
UiT Untitled
 
28 Hansen, Terkel; Ausbacher, Dominik; Zachariassen, Zack Georg; Anderssen, Trude; Havelkova, Martina; Strøm, Morten B..
Anticancer activity of small amphipathic β2,2-amino acid derivatives. European Journal of Medicinal Chemistry 2012 ;Volum 58. s. 22-29
UiT Untitled
 
29 Pohjala, Leena; Ausbacher, Dominik; Strøm, Morten B.; Vuorela, Pia M..
Inhibition of Chlamydia pneumoniae infectivity by β-amino acid derivatives mimicking cationic antimicrobial peptides. 7th meeting of the European society for Chlamydia research; 2012-07-01 - 2012-07-06
UiT Untitled
 
30 Tørfoss, Veronika; Ausbacher, Dominik; Cavalcanti Jacobsen, Cristiane de Albuquerque; Hansen, Terkel; Brandsdal, Bjørn Olav; Havelkova, Martina; Strøm, Morten B..
Synthesis of anticancer heptapeptides containing a unique lipophilic β2,2-amino acid building block. Journal of Peptide Science 2012 ;Volum 18.(3) s. 170-176
UiT Untitled
 
31 Tørfoss, Veronika; Isaksson, Johan; Ausbacher, Dominik; Brandsdal, Bjørn Olav; Flaten, Gøril Eide; Anderssen, Trude; Cavalcanti Jacobsen, Cristiane de Albuquerque; Havelkova, Martina; Nguyen, Leonard T.; Vogel, Hans J.; Strøm, Morten B..
Improved anticancer potency by head-to-tail cyclization of short cationic anticancer peptides containing a lipophilic b2,2-amino acid. Journal of Peptide Science 2012 ;Volum 18.(10) s. 609-619
UiT Untitled
 
2011
32 Ausbacher, Dominik; Hansen, Terkel; Svineng, Gunbjørg; Strøm, Morten B..
Mechanisms of cancer cell death induced by two novel cationic beta-peptidomimetics. Biopolymers 2011 ;Volum 96.(4) s. 456-457
UiT Untitled
 
33 Ausbacher, Dominik; Hansen, Terkel; Svineng, Gunbjørg; Strøm, Morten B..
Mechanisms of cancer cell death induced by two novel cationic β-peptidomimetics. American Peptide Symposium; 2011-06-25 - 2011-06-30
UiT Untitled
 
34 Hansen, Terkel; Ausbacher, Dominik; Flaten, Gøril Eide; Havelkova, Martina; Strøm, Morten B..
Synthesis of Cationic Antimicrobial beta(2,2)-Amino Acid Derivatives with Potential for Oral Administration. Journal of Medicinal Chemistry 2011 ;Volum 54.(3) s. 858-868
UiT Untitled
 
2010
35 Hupfeld, Stefan; Moen, Helene; Ausbacher, Dominik; Haas, Heinrich; Brandl, Martin.
Liposome fractionation and size analysis by asymmetrical flow field-flow fractionation/multi-angle light scattering: influence of ionic strength and osmotic pressure of the carrier liquid. Chemistry and Physics of Lipids 2010 ;Volum 163.(2) s. 141-147
UiT Untitled
 
36 Hansen, Terkel; Ausbacher, Dominik; Havelkova, Martina; Strøm, Morten B..
Bactericidal activity of small β-peptidomimetics. European Peptide Symposium; 2010-09-05 - 2010-09-09
UiT Untitled
 
2009
37 Hupfeld, Stefan; Ausbacher, Dominik; Brandl, Martin.
Asymmetric flow field-flow fractionation of liposomes: 2. Concentration detection and adsorptive loss phenomena. Journal of Separation Science 2009 ;Volum 32.(20) s. 3555-3561
UiT Untitled
 
38 Hupfeld, Stefan; Ausbacher, Dominik; Brandl, Martin.
Asymmetric flow field-flow fractionation of liposomes: optimization of fractionation variables. Journal of Separation Science 2009 ;Volum 32.(9) s. 1465-1470
UiT Untitled